MRGPRX1 agonist 1 [2377379-39-8]
HY-130118
CAS Number2377379-39-8
Product group Chemicals
Estimated Purity99.95
Molecular Weight435.50
Overview
- SupplierMedChem Express
- Product NameMRGPRX1 agonist 1 [2377379-39-8]
- Delivery Days Customer10
- CAS Number2377379-39-8
- CertificationResearch Use Only
- Estimated Purity99.95
- Molecular FormulaC23H21N3O4S
- Molecular Weight435.50
- Scientific DescriptionMRGPRX1 agonist 1 is a highly potent MRGPRX1 agonist (EC50=50 nM) with greater than 50-fold selectivity for delta, micro, and kappa opioid receptors. MRGPRX1 agonist 1 is inactive against MRGPRC11. MRGPRC11 inhibits high voltage-activated (HVA) Ca2+ currents, reduces neurotransmitter release, and mitigates nociceptive transmission in the spinal cord. MRGPRX1 agonist 1 is useful for the study of chronic pain, especially neuropathic pain[1].
- SMILESO=S(C1=CC=CC=C1OC)(NC2=CC=C(C)C=C2OC3=CC4=C(C(N)=NC=C4)C=C3)=O
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200
MSDS
Related products
![MRGPRX1 agonist 1 [2377379-39-8]](https://www.targetmol.com/group3/M00/35/FF/CgoaEGayM6SEd22WAAAAAO7JPPY820.png)
Product group Chemicals
CAS Number2377379-39-8
Estimated Purity99.59%
Molecular Weight435.5
- SizePrice
Product group Chemicals
MRGPRX1 agonist 1ORB1309392
CAS Number2377379-39-8
Estimated Purity99.59%
Molecular Weight435.5
- SizePrice