MRS2365 [436847-09-5]

MedChem Express

MRS2365 [436847-09-5]

10

436847-09-5

Research Use Only

C13H19N5O9P2S

483.33

MRS2365 is a potent and selective P2Y1 receptor (EC50=0.4 nM) /[35S]GTPgammaS binding/beta-arrestin 2 recruitment agonist with an EC50 of 0.4 nM. MRS2365 relieves mechanical allodynia and increases mechanical sensitivity. MRS2365 shows little agonist or antagonist activity at the P2Y12 or P2Y13 receptors[1][2][3][4].

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