MT-802

Biorbyt

MT-802 [2231744-29-7]

10

2231744-29-7

Research Use Only

C41H41N9O8

787.8197486

MT-802 (MT802) is a potent BTK PROTAC that induces degradation of both wild-type and C481S mutant BTK (DC50=9.1 nM).

O(C([H])([H])C([H])([H])OC([H])([H])C(N([H])C1C([H])=C([H])C2=C(C=1[H])C(N(C2=O)C1([H])C(N([H])C(C([H])([H])C1([H])[H])=O)=O)=O)=O)C([H])([H])C([H])([H])N1C([H])([H])C([H])([H])C([H])(C([H])([H])C1([H])[H])N1C2C(=C(N([H])[H])N=C([H])N=2)C(C2C([H])=C([H])C(=C([H])C=2[H])OC2C([H])=C([H])C([H])=C([H])C=2[H])=N1

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