Navafenterol (saccharinate) [1648550-37-1]

MedChem Express

Navafenterol (saccharinate) [1648550-37-1]

10

1648550-37-1

Research Use Only

C45H47N7O9S3

926.09

Navafenterol (AZD-8871) saccharinate is an inhaled dual-acting, potent, selective, and long-lasting M3-antagonist/beta2-agonist (MABA) with long-lasting effects and favorable safety profile. The pIC50 is 9.5 for human M3 receptor, and the pEC50 is 9.5 for beta2-adrenoceptor. Navafenterol saccharinate can be used for the research of chronic obstructive pulmonary disease (COPD). Bronchoprotective and antisialagogue effects. Favorable cardiovascular profile[1].

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