![NEO2734 [2081072-29-7] NEO2734 [2081072-29-7]](https://www.targetmol.com/group3/M00/36/0A/CgoaEGayNOOEbmONAAAAAPld1D8305.png)
NEO2734 [2081072-29-7]
T8658
CAS Number2081072-29-7
Product group Chemicals
Estimated Purity98.56%
Molecular Weight435.44
Overview
- SupplierTargetMol Chemicals
- Product NameNEO2734 [2081072-29-7]
- Delivery Days Customer9
- CAS Number2081072-29-7
- CertificationResearch Use Only
- Chemical NameNEO2734
- Estimated Purity98.56%
- Molecular FormulaC22H24F3N3O3
- Molecular Weight435.44
- Scientific DescriptionNEO2734 (EP31670) is an orally active, selective inhibitor of p300/CBP and BET bromodomains, with an IC50 of less than 30 nM for both targets.
- Shelf life instruction3 years
- SMILESCc1cc(cn(C)c1=O)-c1ccc2nc(C3CCOCC3)n(CCOC(F)(F)F)c2c1
- Storage Instruction-20°C
- UNSPSC12352200
References
- Yan Y, Ma J, Wang D, et al. The novel BET-CBP/p300 dual inhibitor NEO2734 is active in SPOP mutant and wild-type prostate cancer. EMBO Mol Med. 2019,11(11):e10659. doi: 10.15252/emmm.201910659Read this paper