[Nle20] H4 peptide (16-23) [2042178-19-6]

TargetMol Chemicals

[Nle20] H4 peptide (16-23) [2042178-19-6]

9

[Nle20] H4 peptide (16-23) is a potent inhibitor of the histone methyltransferase SETD8, exhibiting strong inhibitory activity (Kd = 0.14 microM) by competing for the substrate binding site on SETD8, thereby inhibiting its methylation of histone H4. This peptide can serve as a lead compound in anticancer therapy.

-20°C

12352202