NNC052090 [184845-43-0]

TargetMol Chemicals

NNC052090 [184845-43-0]

72

184845-43-0

Research Use Only

NNC052090

C27H30N2O2

414.54

NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 microM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at alpha1- and D2-receptors with IC50 values are 266 and 1632 nM respectively.

3 years

C(CCN1CCC(O)(CC1)C2=C(OC)C=CC=C2)N3C=4C(C=5C3=CC=CC5)=CC=CC4

-20°C

12352200