NRA-0160

MedChem Express

NRA-0160 [204718-47-8]

10

204718-47-8

Research Use Only

C24H23F2N3OS

439.52

NRA-0160 is a selective dopamine D4 receptor antagonist, with a K i value of 0.48 nM and with negligible affinity for dopamine D2 receptor ( K i : >10000 nM), D3 receptor ( K i : 39 nM), rat 5-HT2A receptor ( K i : 180 nM) and rat alpha1 adrenoceptor ( K i : 237 nM).

O=C(C1=NC(C2=CC=C(F)C=C2)=C(CCN3CC/C(CC3)=C\C4=CC=CC(F)=C4)S1)N

12352200