Olinone

Biorbyt

Olinone [1770789-37-1]

10

1770789-37-1

Research Use Only

C17H21N3O2

299.3675

Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively, shows high selectivity over BET BRD2 (Kd>300 uM).

O=C1C2C3=C([H])C([H])=C([H])C([H])=C3N(C([H])([H])C([H])([H])C([H])([H])C([H])([H])N([H])C(C([H])([H])[H])=O)C=2C([H])([H])C([H])([H])N1[H]

12352200