Bio-Connect

Palosuran (hydrochloride) [2469274-58-4]

HY-10655A
MedChem Express
CAS Number2469274-58-4
Product group Chemicals
Estimated Purity98.67
Molecular Weight454.99
Sign in to order and to see your custom pricing.
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    Palosuran (hydrochloride) [2469274-58-4]
  • Delivery Days Customer
    10
  • CAS Number
    2469274-58-4
  • Certification
    Research Use Only
  • Estimated Purity
    98.67
  • Molecular Formula
    C25H31ClN4O2
  • Molecular Weight
    454.99
  • Scientific Description
    Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats[1][2].
  • SMILES
    OC(CC1=CC=CC=C1)(CC2)CCN2CCNC(NC3=CC(C)=NC4=CC=CC=C34)=O.[H]Cl
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200