Bio-Connect

PDHK-IN-5

HY-146554
MedChem Express
Molecular Weight493.60
Product group Chemicals
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Overview

  • Supplier
    MedChem Express
  • Product Name
    PDHK-IN-5
  • Delivery Days Customer
    10
  • Certification
    Research Use Only
  • Molecular Formula
    C30H31N5O2
  • Molecular Weight
    493.60
  • Scientific Description
    PDHK-IN-5 (Compound 19) is a potent inhibitor of PDHK with IC50s of 0.006 and 0.0329 microM for PDHK2 and PDHK4, repectively. Pyruvate dehydrogenase kinases (PDHKs) are fascinating agent targets for numerous diseases, including diabetes and cancers. PDHK-IN-5 has the potential for the research of cancer diseases[1].
  • SMILES
    CC1=NC2=C(C3=CC=CC(C4CC4)=C3N2)C=C1C5=NN=C(O5)C(C(C)C)CC(NCC6=CC=CC=C6)=O
  • UNSPSC
    12131703