PF 429242 [947303-87-9]

TargetMol Chemicals

PF 429242

9

947303-87-9

Chemical

Research Use Only

PF 429242

99.27%

C25H35N3O2

409.56

PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 microM). It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 microM).

3 years

N(C(=O)C1=CC=C(CN(CC)CC)C=C1)(CCC2=C(OC)C=CC=C2)[C@@H]3CCNC3

-20°C

12352200