Pictilisib (dimethanesulfonate)

MedChem Express

Pictilisib (dimethanesulfonate) [957054-33-0]

10

957054-33-0

Research Use Only

99.72

C25H35N7O9S4

705.85

Pictilisib dimethanesulfonate (GDC-0941 dimethanesulfonate) is a potent inhibitor of PI3Kalpha/delta with IC50 of 3 nM, with modest selectivity against p110beta (11-fold) and p110gamma (25-fold).

O=S(N1CCN(CC1)CC2=CC3=C(S2)C(N4CCOCC4)=NC(C5=CC=CC6=C5C=NN6)=N3)(C)=O.O=S(O)(C)=O.O=S(O)(C)=O

2°C to 8°C

12352200