Pilaralisib

MedChem Express

Pilaralisib [934526-89-3]

10

934526-89-3

Research Use Only

99.14

C25H25ClN6O4S

541.02

Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kalpha, PI3Kbeta, PI3Kgamma, and PI3Kdelta.

CC(C)(N)C(NC1=CC=CC(S(=O)(NC2=NC3=CC=CC=C3N=C2NC4=CC(OC)=CC=C4Cl)=O)=C1)=O

-20°C,2°C to 8°C

12352200