R 50595 (hydrochloride) [104860-61-9]
HY-115375
CAS Number104860-61-9
Product group Chemicals
Molecular Weight594.52
Overview
- SupplierMedChem Express
- Product NameR 50595 (hydrochloride) [104860-61-9]
- Delivery Days Customer9
- CAS Number104860-61-9
- CertificationResearch Use Only
- Molecular FormulaC30H35Cl2F2N3O3
- Molecular Weight594.52
- Scientific Description50595 hydrochloride is a selective noncompetitive cisapride antagonist that interferes with the activity of cisapride and BRL 24924. R 50595 hydrochloride has no effect on the response to electrical stimulation at concentrations up to 3 X 10(-7) M. R 50595 hydrochloride antagonizes the effects of cisapride and BRL 24924 in a noncompetitive manner. R 50595 hydrochloride completely abolishes the effects of 5-HT at a concentration of 3 X 10(-7) M and also antagonizes the effects of 5-HT in a noncompetitive manner[1].
- SMILESO=C(N[C@@H]1[C@@H](OC)CN(CCCC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3)CC1)C4=CC(Cl)=C(N)C=C4OC.[H]Cl
- UNSPSC12352200