(R)-I-BET762 carboxylic acid

MedChem Express

(R)-I-BET762 carboxylic acid

5

Research Use Only

99.50

C20H17ClN4O3

396.83

(R)-I-BET762 carboxylic acid, the R-enantiomer of I-BET762 carboxylic acid (HY-107443). I-BET762 carboxylic acid is an I-BET762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. I-BET762 carboxylic acid is a BRD4 inhibitor with a pIC50 value of 5.1[1].

CC1=NN=C2[C@@H](CC(O)=O)N=C(C3=CC=C(Cl)C=C3)C4=C(C=CC(OC)=C4)N21

-20°C,2°C to 8°C

12352200