rel-A-395 (hydrochloride)
HY-101512D
Molecular Weight523.11
Product group Chemicals
Overview
- SupplierMedChem Express
- Product Namerel-A-395 (hydrochloride)
- Delivery Days Customer999
- CertificationResearch Use Only
- Molecular FormulaC26H36ClFN4O2S
- Molecular Weight523.11
- Scientific Descriptionrel-A-395 hydrochloride is the relative configuration of A-395 (HY-101512) hydrochloride. A-395 is an antagonist of polycomb repressive complex 2 (PRC2) protein-protein interactions that potently inhibits the trimeric PRC2 complex (EZH2-EED-SUZ12) with an IC50 of 18 nM[1].
- SMILESO=S(N1CCN(C2=CC=C([C@H]3CN(C4C(C(F)=CC=C5)=C5CC4)C[C@@H]3N(C)C)C=C2)CC1)(C)=O.Cl
- UNSPSC12352200