Relacorilant [1496510-51-0]

TargetMol Chemicals

Relacorilant [1496510-51-0]

9

Chemical

Research Use Only

Relacorilant

98.99%

C27H22F4N6O3S

586.56

Relacorilant is a selective and orally bioavailable antagonist of glucocorticoid receptor(Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively). Relacorilant has the potential for Cushings syndrome treatment.

3 years

C(=O)([C@@]12C(=CC3=C(C1)C=NN3C4=CC=C(F)C=C4)CCN(S(=O)(=O)C5=CN(C)N=C5)C2)C6=CC(C(F)(F)F)=CC=N6

-20°C

12352200