Ritanserin [87051-43-2]

MedChem Express

Ritanserin [87051-43-2]

10

87051-43-2

Research Use Only

99.78

C27H25F2N3OS

477.57

Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic alpha1, Adrenergic alpha2 receptors[1].

CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5

-20°C

12352200