Rolapitant (Standard) [552292-08-7]

MedChem Express

Rolapitant (Standard) [552292-08-7]

5

552292-08-7

CHEMICAL,detergents_surfactants

Research Use Only

500.48

Rolapitant (Standard) is the analytical standard of Rolapitant. This product is intended for research and analytical applications. Rolapitant (SCH619734) is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a Ki of 0.66 nM. Rolapitant does not interact with CYP3A4. Rolapitant shows potent anti-emetic activity in a ferret emesis model[1][2].

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12352005