RS-127445

MedChem Express

RS-127445 [199864-87-4]

5

199864-87-4

Research Use Only

99.62

C17H16FN3

281.33

RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites[1].

NC1=NC(C(C)C)=CC(C2=C3C=CC=CC3=C(F)C=C2)=N1

2°C to 8°C

12352200