(S)-(+)-Dimethindene (maleate) [136152-65-3]
HY-107647
CAS Number136152-65-3
Product group Chemicals
Estimated Purity99.94
Molecular Weight408.49
Overview
- SupplierMedChem Express
- Product Name(S)-(+)-Dimethindene (maleate) [136152-65-3]
- Delivery Days Customer10
- CAS Number136152-65-3
- CertificationResearch Use Only
- Estimated Purity99.94
- Molecular FormulaC24H28N2O4
- Molecular Weight408.49
- Scientific Description(S)-(+)-Dimethindene maleate, an enantiomer, is a potent M2-selective muscarinic receptor antagonist (pA2 = 7.86/7.74; pKi = 7.78). (S)-(+)-Dimethindene maleate shows lower affinities for the muscarinic M1 (pA2 = 6.83/6.36; pKi = 7.08), the M3 (pA2 = 6.92/6.96; pKi = 6.70) and the M4 receptors (pKi = 7.00), respectively. (S)-(+)-Dimethindene maleate also is a histamine H1 receptor antagonist (pA2 = 7.48)[1].
- SMILESC[C@@H](C1=C(CCN(C)C)CC2=C1C=CC=C2)C3=NC=CC=C3.OC(/C=C\C(O)=O)=O
- Storage Instruction2°C to 8°C
- UNSPSC12352200
![(S)-(+)-Dimethindene maleate [136152-65-3]](https://www.targetmol.com/group3/M00/36/15/CgoaEGayNzGEfEkxAAAAAC57emo131.png)