S1RA (hydrochloride)
HY-18099A
CAS Number1265917-14-3
Product group Chemicals
Estimated Purity99.94
Molecular Weight373.88
Overview
- SupplierMedChem Express
- Product NameS1RA (hydrochloride) [1265917-14-3]
- Delivery Days Customer9
- CAS Number1265917-14-3
- CertificationResearch Use Only
- Estimated Purity99.94
- Molecular FormulaC20H24ClN3O2
- Molecular Weight373.88
- Scientific DescriptionS1RA (E-52862) hydrochloride is an orally active and selective sigma-1 receptor (sigma1R) antagonist with a Ki value of 17 nM. S1RA hydrochloride shows good selectivity against sigma2R (Ki >1000 nM). S1RA hydrochloride is a human 5-HT2B receptor antagonist with an IC50 value of 4.7 microM. S1RA hydrochloride inhibits neuropathic pain and activity-induced spinal sensitization[1][2].
- SMILESCC1=CC(OCCN2CCOCC2)=NN1C3=CC(C=CC=C4)=C4C=C3.[H]Cl
- Storage Instruction2°C to 8°C
- UNSPSC12352200
Related products
![S1RA hydrochloride [1265917-14-3]](https://www.targetmol.com/group3/M00/37/ED/CgoaEGayU8SEegSpAAAAAKnB7q8050.png)
Product group Chemicals
CAS Number1265917-14-3
Estimated Purity99.65%
Molecular Weight373.87
- SizePrice
Product group Chemicals
S1RA hydrochlorideORB1303040
CAS Number1265917-14-3
Estimated Purity99.78%
Molecular Weight373.87
- SizePrice
Product group Chemicals
S1RA hydrochlorideBS177543
CAS Number1265917-14-3
Molecular Weight373.88 g/mol
- SizePrice
