Saclofen
HY-100813
CAS Number125464-42-8
Product group Chemicals
Estimated Purity99.87
Molecular Weight249.719
Overview
- SupplierMedChem Express
- Product NameSaclofen [125464-42-8]
- Delivery Days Customer10
- CAS Number125464-42-8
- Estimated Purity99.87
- Molecular FormulaC9H12ClNO3S
- Molecular Weight249.719
- Scientific DescriptionSaclofen is an orally available competitive GABA B receptor antagonist with an IC 50 of 7.8 microM, but it has a weaker antagonistic effect on GABA B1b and GABA B2 heterodimer recombinant receptors. Saclofen can inhibit the binding of baclofen (HY-B007) to rat cerebellar membranes and block the phase shifts in circadian rhythms caused by baclofen. Saclofen has also shown anti-inflammatory and analgesic effects in rats [1] [2] [3] [4] [5] .
- SMILESO=S(CC(CN)C1=CC=C(Cl)C=C1)(O)=O
- Storage Instruction-20°C
- UNSPSC12352200