Bio-Connect

Samelisant

HY-120124
MedChem Express
CAS Number1394808-20-8
Product group Chemicals
Estimated Purity98.65
Molecular Weight446.41
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Samelisant [1394808-20-8]
  • Delivery Days Customer
    10
  • Applications
    ELISA
  • CAS Number
    1394808-20-8
  • Certification
    Research Use Only
  • Estimated Purity
    98.65
  • Molecular Formula
    C21H33Cl2N3O3
  • Molecular Weight
    446.41
  • Scientific Description
    Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability. Samelisant has a similar binding affinity towards human (hH3R; K i =8.7 nM) and rat (rH3R;K i =9.8 nM) H3R indicating no inter-species differences. Samelisant can be used for the research of sleep-related disorders [1] .
  • SMILES
    O=C(CN1CCOCC1)NC2=CC=C(C=C2)OC3CCN(CC3)C4CCC4.[H]Cl.[H]Cl
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200