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Samuraciclib (hydrochloride)

HY-103712A
MedChem Express
CAS Number1805789-54-1
DownloadMSDS
Product group Chemicals
Estimated Purity99.98
Molecular Weight430.97
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Samuraciclib (hydrochloride) [1805789-54-1]
  • Delivery Days Customer
    10
  • CAS Number
    1805789-54-1
  • Certification
    Research Use Only
  • Estimated Purity
    99.98
  • Molecular Formula
    C22H31ClN6O
  • Molecular Weight
    430.97
  • Scientific Description
    Samuraciclib hydrochloride (CT7001 hydrochloride) is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC 50 of 41 nM. Samuraciclib hydrochloride displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC 50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib hydrochloride inhibits the growth of breast cancer cell lines with GI 50 values between 0.2-0.3 microM. Samuraciclib hydrochloride has anti-tumor effects [1] [2] .
  • SMILES
    O[C@H]1CNCC[C@@H]1CNC2=NC3=C(C(C)C)C=NN3C(NCC4=CC=CC=C4)=C2.[H]Cl
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200