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Samuraciclib (hydrochloride dihydrate)

HY-103712B
MedChem Express
Estimated Purity99.08
DownloadMSDS
Product group Chemicals
Molecular Weight521.70
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Samuraciclib (hydrochloride dihydrate)
  • Delivery Days Customer
    10
  • Certification
    Research Use Only
  • Estimated Purity
    99.08
  • Molecular Formula
    C22H30N6O.(2.5HCl).(2H2O)
  • Molecular Weight
    521.70
  • Scientific Description
    Samuraciclib (CT7001) hydrochloride hydrate is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC 50 of 41 nM. Samuraciclib hydrochloride hydrate displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC 50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib hydrochloride hydrate inhibits the growth of breast cancer cell lines with GI 50 values between 0.2-0.3 microM. Samuraciclib hydrochloride hydrate has anti-tumor effects [1] [2] .
  • SMILES
    O[C@H]1CNCC[C@@H]1CNC2=NC3=C(C(C)C)C=NN3C(NCC4=CC=CC=C4)=C2.Cl.O.O.[2.5]
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200