Sarpogrelate (hydrochloride) [135159-51-2]

MedChem Express

Sarpogrelate (hydrochloride) [135159-51-2]

10

135159-51-2

Research Use Only

99.09

C24H32ClNO6

465.97

Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, alpha1-, alpha2- and beta-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis[1][2][3].

COC1=CC=CC(CCC2=CC=CC=C2OCC(CN(C)C)OC(CCC(O)=O)=O)=C1.Cl

2°C to 8°C

12352200