SKF-82958 [80751-65-1]

MedChem Express

SKF-82958 [80751-65-1]

10

80751-65-1

Research Use Only

C19H20ClNO2

329.82

SKF-82958 ((+/-)-SKF 82958) is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM)[1].

OC1=C(O)C=C2C(C3=CC=CC=C3)CN(CC=C)CCC2=C1Cl

12352200