SKF-82958 (hydrobromide) (Standard) [74115-01-8]
HY-10435AR
Product group Assays
Overview
- SupplierMedChem Express
- Product NameSKF-82958 (hydrobromide) (Standard) [74115-01-8]
- Delivery Days Customer5
- CertificationResearch Use Only
- Scientific DescriptionSKF-82958 (hydrobromide) (Standard) is the analytical standard of SKF-82958 (hydrobromide). This product is intended for research and analytical applications. SKF-82958 ((+/-)-SKF 82958) hydrobromide is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM)[1].
- UNSPSC41116100