Bio-Connect

SMU-B [1253286-90-6]

HY-120387
MedChem Express
CAS Number1253286-90-6
Product group Chemicals
Molecular Weight515.41
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Overview

  • Supplier
    MedChem Express
  • Product Name
    SMU-B [1253286-90-6]
  • Delivery Days Customer
    5
  • CAS Number
    1253286-90-6
  • Certification
    Research Use Only
  • Molecular Formula
    C26H25Cl2FN4O2
  • Molecular Weight
    515.41
  • Scientific Description
    SMU-B is the orally active inhibitor for ALK (IC50c-ros oncogene 1 (ROS1), c-MET (IC50=1.87 nM) and AXL (IC50=28.9 nM). SMU-B inhibits the proliferation of MKN45, H1993 and H441 with IC50s of 0.02 microM, 1.58 microM and 2.82 microM, respectively. SMU-B exhibits antitumor efficacy in mouse models[1][2].
  • SMILES
    O=C1NC2=C(C=CC(C3=CC(O[C@@H](C4=C(Cl)C=CC(F)=C4Cl)C)=C(N)N=C3)=C2)C15CCN(C)CC5
  • UNSPSC
    12352200