SRA880 malonate

Biorbyt

SRA880 malonate

10

Research Use Only

98.00%

C29H36N4O8

568.62

SRA880 is a non-peptide somatostatin sst(1) receptor antagonist which displays a significantly lower affinity for the other human recombinant somatostatin receptors ( pK(d)= 6.0) or a wide range of neurotransmitter receptors, except for the human dopamine D4 receptors. SRA880 positively modulates the release of endogenous SRIF, was found to synergize with imipramine in causing antidepressant-like effects in the tail suspension test.

C(C(O)=O)C(O)=O.CN1[C@]2([C@@](CC=3C(C2)=CC=CC3OC)(C[C@@H](C(=O)N4CCN(CC4)C5=CC=C(N(=O)=O)C=C5)C1)[H])[H]

-20°C

12352200