SSR240612 [464930-42-5]
HY-15039
CAS Number464930-42-5
Product group Chemicals
Estimated Purity99.51%
Molecular Weight793.41
Overview
- SupplierMedChem Express
- Product NameSSR240612 [464930-42-5]
- Delivery Days Customer10
- CAS Number464930-42-5
- CertificationResearch Use Only
- Estimated Purity99.51%
- Molecular FormulaC42H53ClN4O7S
- Molecular Weight793.41
- Scientific DescriptionSSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist, with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.
- SMILESO=S(N[C@@H](C1=CC=C2C(OCO2)=C1)CC(N[C@@H](C(N(C)C(C)C)=O)CC3=CC=C(CN([C@@H]4C)[C@H](CCC4)C)C=C3)=O)(C5=CC(C=CC(OC)=C6)=C6C=C5)=O.Cl[H]
- Storage Instruction2°C to 8°C,-20°C,-80°C
- UNSPSC12352200