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Sunitinib malate

S1042
Selleck Chemicals
CAS Number341031-54-7
Product group Chemicals
Estimated Purity...
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Sunitinib (SU11248) malate [341031-54-7]
  • Delivery Days Customer
    9
  • CAS Number
    341031-54-7
  • Certification
    Research Use Only
  • Estimated Purity
    ...
  • Scientific Description
    Sunitinib malate is a multi-targeted RTK inhibitor targeting VEGFR2 (Flk-1) and PDGFRbeta with IC50 of 80 nM and 2 nM in cell-free assays, and also inhibits c-Kit. Sunitinib Malate effectively inhibits autophosphorylation of Ire1alpha. Sunitinib Malate increases both death receptor and mitochondrial-dependent apoptosis.
  • Storage Instruction
    -80°C
  • UNSPSC
    51202000

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