Taselisib

MedChem Express

Taselisib [1282512-48-4]

10

1282512-48-4

Research Use Only

99.75

C24H28N8O2

460.53

Taselisib (GDC-0032) is a potent PI3K inhibitor targets PIK3CA mutations, with K i s of 0.12 nM, 0.29 nM, 0.97 nM, and 9.1 nM for PI3Kdelta, PI3Kalpha, PI3Kgamma and PI3Kbeta, respectively.

CC(C)N1C(C2=CN3C(C(C(OCC3)=C4)=CC=C4C5=CN(C(C)(C(N)=O)C)N=C5)=N2)=NC(C)=N1

-20°C,2°C to 8°C

12352200