TC-G 1005

MedChem Express

TC-G 1005 [1415407-60-1]

10

1415407-60-1

Research Use Only

99.83

C25H25N3O2

399.48

TC-G 1005 is a potent, selective and orally active agonist of the BA receptor Takeda G protein-coupled receptor 5 (TGR5) , with EC 50 s of 0.72 and 6.2 nM for hTGR5 and mTGR5, respectively. TC-G 1005 can reduce glucose levels in vivo [1] [2] .

O=C(C1=CN=CC=C1OC2=C(C=CC(C)=C2)C)N3C4=CC=CC=C4N(C5CC5)CC3

-20°C,2°C to 8°C

12352200