Thioperamide (maleate) [148440-81-7]

MedChem Express

Thioperamide (maleate) [148440-81-7]

10

148440-81-7

Research Use Only

98.26

C15H24N4S.xC4H4O4

Thioperamide maleate (MR-12842 maleate) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. Thioperamide maleate inhibits [3H]histamine synthesis with a Ki of 31 nM[1].

S=C(N1CCC(C2=CN=CN2)CC1)NC3CCCCC3.O=C(O)/C=C\C(O)=O.[x]

2°C to 8°C

12352200