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Tofacitinib (CP-690550) [477600-75-2]

S2789
Selleck Chemicals
Product group Chemicals
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Tofacitinib (CP-690550) [477600-75-2]
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Scientific Description
    Tofacitinib (CP-690550,Tasocitinib) is a novel inhibitor of JAK3 with IC50 of 1 nM in cell-free assays, 20- to 100-fold less potent against JAK2 and JAK1. Tofacitinib inhibits the expression of antiapoptotic BCL-A1 and BCL-XL in human plasmacytoid dendritic cells (PDC) and induced PDC apoptosis.
  • UNSPSC
    12352200

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