TP-238 [2415263-04-4]

MedChem Express

TP-238 [2415263-04-4]

10

2415263-04-4

Research Use Only

C22H30N6O3S

458.58

TP-238 is a potent and selective dual CECR2/BPTF probe with IC50 values of 30 nM and 350 nM, respectively. TP-238 also inhibits BRD9 with a pIC50 of 5.9 and is less active against other 338 kinases[1][2].

CN(C)CCCOC1=CC=C(C=C1)C2=CC(NCCCN3N=CC=C3)=NC(S(=O)(C)=O)=N2

12352200