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Tracazolate (hydrochloride) [1135210-68-2]

HY-B1803A
MedChem Express
CAS Number1135210-68-2
Product group Chemicals
Estimated Purity99.24
Molecular Weight340.85
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Tracazolate (hydrochloride) [1135210-68-2]
  • Delivery Days Customer
    10
  • CAS Number
    1135210-68-2
  • Certification
    Research Use Only
  • Estimated Purity
    99.24
  • Molecular Formula
    C16H25ClN4O2
  • Molecular Weight
    340.85
  • Scientific Description
    Tracazolate (ICI 136753) hydrochloride is a potent GABAA receptor modulator. Tracazolate hydrochloride has selectivity for beta3 and potentiates alpha1beta1gamma2s (EC50=13.2 microM), alpha1beta3gamma2 (EC50=1.5 microM). Tracazolate hydrochloride has the potency (EC50) determined by the nature of the third subunit (gamma1-3, delta, epsilon) within the receptor complex. Tracazolate hydrochloride possesses anxiolytic and anticonvulsant activity[1][2].
  • SMILES
    O=C(C1=C(C)N=C(N(CC)N=C2)C2=C1NCCCC)OCC.[H]Cl
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200