UBP316 [936095-50-0]

MedChem Express

UBP316 [936095-50-0]

10

936095-50-0

Research Use Only

99.95

C20H19N3O6S

429.45

UBP316 (ACET) is a highly potent and selective kainate receptor GluK1 (GluR5) antagonist, with a Kb value of 1.4 nM. UBP316 is effective at blocking the depression of both field excitatory postsynaptic potentials (fEPSPs) and monosynaptically-evoked GABAergic transmission induced by ATPA, a GluK1 selective agonist[1].

OC(C(SC(C1=CC=CC=C1)=C2)=C2CN3C(N(C=C(C)C3=O)C[C@H](N)C(O)=O)=O)=O

-20°C,2°C to 8°C

12352200