UMB-32 [1635437-39-6]

TargetMol Chemicals

UMB-32 [1635437-39-6]

44

1635437-39-6

Research Use Only

UMB-32

C21H23N5O

361.44

UMB-32 is a potent and selective BRD4 inhibitor, demonstrating an affinity for BRD4 with a dissociation constant (K d) of 550 nM and an inhibitory concentration 50 (IC 50) of 637 nM. Moreover, UMB-32 exhibits effectiveness against TAF1, a bromodomain-containing transcription factor [1].

3 years

N(C(C)(C)C)C1=C(N=C2N1C=CN=C2)C3=CC=C(C=C3)C=4C(C)=NOC4C

-20°C

12352200