Bio-Connect

UNC10013

HY-173156
MedChem Express
Molecular Weight982.85
Product group Chemicals
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Overview

  • Supplier
    MedChem Express
  • Product Name
    UNC10013
  • Delivery Days Customer
    5
  • Certification
    Research Use Only
  • Molecular Formula
    C37H54F12N8O9
  • Molecular Weight
    982.85
  • Scientific Description
    UNC10013 is a SETDB1 allosteric modulator that forms a covalent bond with Cys385 in the 3TD domain, exhibiting negative allosteric regulatory activity. It has a kinact/KI value of 1.0 x 106 M-1*s-1. UNC10013 effectively disrupts SETDB1-mediated Akt methylation and holds potential value for research in cancer and neurodegenerative diseases.
  • SMILES
    O=C(NC1=CC2=C(NCCCCCCN(C)C)N=C(NCCCCCN(C)C)N=C2C=C1)/C=C/CN(C)C.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F
  • UNSPSC
    12352200