Varenicline (Tartrate) (Standard)
HY-10021R
Product group Assays
Overview
- SupplierMedChem Express
- Product NameVarenicline (Tartrate) (Standard) [375815-87-5]
- Delivery Days Customer5
- CertificationResearch Use Only
- Scientific DescriptionVarenicline (Tartrate) (Standard) is the analytical standard of Varenicline (Tartrate). This product is intended for research and analytical applications. Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agonist of alpha6beta2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].
- UNSPSC41116135