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Vasopressin V2 receptor antagonist 1 [2648650-50-2]

HY-146272
MedChem Express
CAS Number2648650-50-2
Product group Chemicals
Molecular Weight589.12
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Vasopressin V2 receptor antagonist 1 [2648650-50-2]
  • Delivery Days Customer
    10
  • CAS Number
    2648650-50-2
  • Certification
    Research Use Only
  • Molecular Formula
    C33H37ClN4O4
  • Molecular Weight
    589.12
  • Scientific Description
    Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2 receptor (V2R) antagonist with a Ki of 3.8 nM. Vasopressin V2 receptor antagonist 1 can be used for autosomal dominant polycystic kidney disease (ADPKD) research[1].
  • SMILES
    ClC1=CC2=C(C=C1)N(C(C3=C(C=C(C=C3)NC(C4=C(C=CC=C4)C)=O)C)=O)CCCC2NCCC(N5CCOCC5)=O
  • UNSPSC
    12131703