Velusetrag (hydrochloride) [866933-51-9]

MedChem Express

Velusetrag (hydrochloride) [866933-51-9]

10

866933-51-9

Research Use Only

98.95

C25H37ClN4O5S

541.10

Velusetrag (TD-5108) hydrochloride is an orally active, potent and selective agonist of serotonin 5-HT4 receptor (5-HT4R), with a pKi of 7.7. Velusetrag hydrochloride exhibits no affinity (Ki>10 microM) for 5-HT2A and 5-HT2B receptors. Velusetrag hydrochloride can be used for the research of gastrointestinal diseases and Parkinsons disease[1][2][3][4][5].

[H]Cl.O=C(C1=CC2=C(N(C(C)C)C1=O)C=CC=C2)N[C@@H]3C[C@@H](N4C[C@@H](O)CN(C)S(=O)(C)=O)CC[C@@H]4C3

2°C to 8°C

12352200