VPC-3033 [110763-24-1]
HY-118409
CAS Number110763-24-1
Product group Chemicals
Molecular Weight298.33
Overview
- SupplierMedChem Express
- Product NameVPC-3033 [110763-24-1]
- Delivery Days Customer9
- CAS Number110763-24-1
- CertificationResearch Use Only
- Molecular FormulaC21H14O2
- Molecular Weight298.33
- Scientific DescriptionVPC-3033 is an androgen receptor antagonist. VPC-3033 has a strong androgen DHT replacement potency (IC50: 0.625-2.5 microM), can effectively inhibit androgen receptor transcriptional activity (IC50=0.3 microM), and has a strong androgen receptor degradation ability. In addition, VPC-3033 exhibits significant anti-androgen receptor activity against prostate cancer cells resistant to Enzalutamide (HY-70002)[1].
- SMILESO=C1C2=C(/C(C3=C1C=CC=C3)=C\C4=CC(O)=CC=C4)C=CC=C2
- UNSPSC12352200