Bio-Connect

VU0152099 [612514-42-8]

HY-119226
MedChem Express
CAS Number612514-42-8
Product group Chemicals
Estimated Purity98.25
Molecular Weight355.41
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Overview

  • Supplier
    MedChem Express
  • Product Name
    VU0152099 [612514-42-8]
  • Delivery Days Customer
    10
  • CAS Number
    612514-42-8
  • Certification
    Research Use Only
  • Estimated Purity
    98.25
  • Molecular Formula
    C18H17N3O3S
  • Molecular Weight
    355.41
  • Scientific Description
    VU0152099 is a potent, selective and brain-penetrant mAChR M4 positive allosteric modulator with an EC50 of 0.4 microM for rat M4 receptor. VU0152099 is inactive for other mAChR subtypes or other GPCRs. VU0152099 has no agonist activity but potentiated responses of M4 to acetylcholine[1].
  • SMILES
    O=C(C1=C(N)C2=C(C)C=C(C)N=C2S1)NCC3=CC=C(OCO4)C4=C3
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200