WAY-100635 maleate

Biorbyt

WAY-100635 maleate

16

634908-75-1

Research Use Only

C29H38N4O6

538.6352

WAY-100635 is a potent, silent antagonist of 5-HT1A receptors (IC50 = 2.2 nM; Ki = 0.84 nM for rat 5-HT1A receptors). Displays 100-fold selectivity for 5-HT1A over other 5-HT subtypes. Also exhibits agonist activity at dopamine D4 receptors.

OC(/C=C\C(=O)O)=O.COC1=CC=CC=C1N1CCN(CCN(C(C2CCCCC2)=O)C2=CC=CC=N2)CC1

12352200