YM-58790 [214558-72-2]

MedChem Express

YM-58790 [214558-72-2]

10

214558-72-2

Research Use Only

98.21

C27H32ClN3O2

466.01

YM-58790 is a potent antagonist of mAChR. YM-58790 binds M1, M2, M3 with Ki values of 28 nM, 260 nM, and 15 nM. YM-58790 exhibits potent inhibitory activity on bladder pressuer in reflexly-evoked rhythmic contraction in rats[1].

O=C(OC1CCN(CC2=CC=C(NC)C=C2)CC1)NC(C3=CC=CC=C3)C4=CC=CC=C4.[H]Cl

2°C to 8°C

12352200